Raukawa Rawa Raukawa 7P (1890208-58-8) ataata
Raukawa Rawa 7P (1890208-58-8) Whakaahuatanga
Ko te konupae Rawa 7P e whakatairanga ana i te tipu o te koiora tuatahi mai i te hippocampus, te cortex, me te retina. i roto i te tauira kararehe o te whara nerve opic, Kua whakaatuhia te paura 7P Hangarau ki te whakatipu i te tipu o te aukati-43 pai axons, tohu e te mahi i roto i te vitiviti o te Raw Compound 7P paura whakawhiti ki te whakaongaonga o te whakaoranga axon i roto i vivo.further arotakenga o Ko te Hangarau Rawa 7P te paura me te whakawhitinga ake o nga hanga e hangaia ai te whakaora i roto i te vivon i roto i te ora, ka whakaratohia he kaupapa whaanui mo nga mahi ki te whakarei ake i nga rautaki maimoatanga.
raw 2 - [(2-methoxyphenyl) [(4-methyl phenyl) sulfonyl] amino] -N- (4-methoxy-3-pyridinyl) acetamide (Hua 7P) paura (1890208-58-8) Snga whakaritenga
ingoa hua | 2 - [(2-methoxyphenyl) [(4-methyl phenyl) sulfonyl] amino] -N- (4-methoxy-3-pyridinyl) acetamide (Paahana 7P Raw) |
Ingoa Toi | 2 - [(2-methoxyphenyl) [(4-methyl phenyl) sulfonyl] amino] -N- (4-methoxy-3-pyridinyl) acetamide (Raw Compound 7P paura) |
Brand Name | Raukawa Rawa 7P |
Kaupapa Drug | Nootropic Drugs |
CAS Tau | 1890208-58-8 |
INCHIKey | NAXWKPFXCOBXLE-UHFFFAOYSA-N |
rāpoi FTuhinga | C22H23N3O5S |
rāpoi Wwaru | 441.508g |
Ko te Monoisotopic Mass | 440G / mol |
ira whakakoero | N / He |
Fwhakahou Phinu | N / He |
Hawhe-Haiao-Ora | N / He |
Tae | paura White |
STuhinga | paku pakuhia i roto i te wai me te waihano. |
Stora Tte taumaha | Whakaorangia i te pāmahana rūma, i te hiri hiri, ka karo i te wera kaha me te marama. |
Apātai | • Te whakanui ake i te whakaritenga • Whakapai ake i te taiao • Awhina i te ngoikoretanga whawhai • Aukati i te waikura i roto i te roro • Ka pangia te waipiro o te roro |
raw Putanga 7P puehu (1890208-58-8) Whakaahuatanga
Pūhui Katoa 7P (2 - [(2-methoxyphenyl) [(4-methyl phenyl) sulfonyl] amino] -N- (4-methoxy-3-pyridinyl) acetamide) puehu e whakatairanga ana i te tipu neurite o nga neuron tuatahi ahurea i ahu mai i te hippocampus , uho roro, me te retina. i roto i te tauira kararehe o te whara nerve whatu, i whakaatuhia te Raw Compound 7P paura hei whakatipu tipu o te haangai-43 pai o te haakona, e tohu ana ko te ngoikoretanga in vitro i te tipu o te Raw Powhao 7P paura ka huri hei whakaohooho i te whakahou i te toki i roto i te vivo. Ko te Paura Miihini 7P paura me te whakamarama i nga tikanga e taea ai te whakahou i te haaka i roto i te waa ka whakarato i te kaupapa whaitake mo nga mahi a meake nei ki te whakarei ake i nga rautaki maimoatanga.
Whakamahia te 7P Hanga puehu (1890208-58-8)
Ko te 7p (2 - [(2-methoxyphenyl) [[4-methyl phenyl] sulfonyl] amino] -N- (4-methoxy-3-pyridinyl) acetamide) i whakaatu i te mahi tino nui ki nga moenga pukupuku pukupuku. I roto i te tauira ngutu o te kiore i hangaia me nga waehu HeLa, i whakaatu te 7p i te waihanga o te whanaketanga pukupuku o te pukupuku o te pukupuku. Ko te whakamätautau ä-hitori o te rorohiko e whakaatuhia ana e te 7p te whakapai ake i te microstructure i roto i te tikanga toenga-teitei. I whakanui ano te 7p i te nui o nga waehu HeLa i roto i te G0 / G1 me te S-waa, a ka whakaiti rawa i te waahanga o te G2 / M-phase. Ko nga hua o 7p i runga i te C-caspase-3, C-caspase-9, Bcl-2 me te korero Bax i roto i nga waehu HeLa i whakatau hoki.
Ko te whakatairanga polymerization o te tubulin, he rangahau mo te immunofluorescence, te rangahau huringa o te taiao, me te whakamatau whakataetae tubulin-whakataetae whakataetae kua kaha te whakaatu ko te 7p he kaitautoko o te kohinga o te tubulin.
painga of Putanga 7P puehu (1890208-58-8)
I whakatairanga te 7p ki te whakahou i te whakaoranga o te matapihi
Whakahokia te mahunga o te kino
tūtohu Putanga 7P puehu (1890208-58-8) Tauranga
I whakaatuhia e 7p te 100% te inhibition o te parasitemia i te ra 4 i nga doses maha (100, 50, me te 25 mg / kg) kua hoatu mo nga ra e wha, engari i te 100 mg / kg, ka ora nga kiore katoa, ka ora, i te 50 mg / kg, e toru o nga kiore e rima i ora, e rua nga kiore i ora, i te 25 mg / kg, kaore tetahi o nga kiore i ora